Roundtable Discussion: Into the Thick of It: Oligonucleotides into the Brain with Depth, Precision & Safety

  • Achieving deep brain oligonucleotide exposure while managing acute and chronic neurotoxicity
  • The role of imaging and PK/PD modelling in optimising CNS dosing strategies
  • Limitations of transferrin receptor-mediated delivery and emerging alternative shuttle approaches
  • Balancing regional coverage, cell-type specificity, and peripheral exposure risks
  • Translational and safety considerations impacting clinical development and regulatory confidence